British Journal of Pharmacology

Second M₃ muscarinic receptor binding site contributes to bronchoprotection by tiotropium

Pages: 2864-2876

Article date: August 2019

Authors: Loes E.M. Kistemaker, Carolina R.S. Elzinga, Christofer S. Tautermann, Michael P. Pieper, Daniel Seeliger, Suraya Alikhil, Martina Schmidt, Herman Meurs, Reinoud Gosens

A photoswitchable GABA receptor channel blocker

Pages: 2661-2677

Article date: August 2019

Authors: Galyna Maleeva, Daniel Wutz, Karin Rustler, Alba Nin‐Hill, Carme Rovira, Elena Petukhova, Antoni Bautista‐Barrufet, Alexandre Gomila‐Juaneda, Petra Scholze, Franck Peiretti, Mercedes Alfonso‐Prieto, Burkhard König, Pau Gorostiza, Piotr Bregestovski

Molecular dynamics simulations of dihydro‐β‐erythroidine bound to the human α4β2 nicotinic acetylcholine receptor

Pages: 2750-2763

Article date: August 2019

Authors: Rilei Yu, Han‐Shen Tae, Qingliang Xu, David J. Craik, David J. Adams, Tao Jiang, Quentin Kaas

Ursodeoxycholic acid accelerates bile acid enterohepatic circulation

Pages: 2848-2863

Article date: August 2019

Authors: Yunjing Zhang, Runqiu Jiang, Xiaojiao Zheng, Sha Lei, Fengjie Huang, Guoxiang Xie, Sandi Kwee, Herbert Yu, Christine Farrar, Beicheng Sun, Aihua Zhao, Wei Jia

Bouchardatine analogue alleviates non‐alcoholic hepatic fatty liver disease/non‐alcoholic steatohepatitis in high‐fat fed mice by inhibiting ATP synthase activity

Pages: 2877-2893

Article date: August 2019

Authors: Yong Rao, Yu‐Ting Lu, Chan Li, Qin‐Qin Song, Yao‐Hao Xu, Zhao Xu, Yu‐Tao Hu, Hong Yu, Lin Gao, Lian‐Quan Gu, Ji‐Ming Ye, Zhi‐Shu Huang

Inhibitors of DAG metabolism suppress CCR2 signalling in human monocytes

Pages: 2736-2749

Article date: August 2019

Authors: Priscilla Day, Lisa Burrows, David Richards, Samuel J. Fountain

Selected Abstracts from Pharmacology 2018

Pages: 2977-3081

Article date: August 2019

Glucagon up‐regulates hepatic mitochondrial pyruvate carrier 1 through cAMP‐responsive element‐binding protein; inhibition of hepatic gluconeogenesis by ginsenoside Rb1

Pages: 2962-2976

Article date: August 2019

Authors: Meng‐Die Lou, Jia Li, Yao Cheng, Na Xiao, Gaoxiang Ma, Ping Li, Baolin Liu, Qun Liu, Lian‐Wen Qi

Acute activation of endothelial AMPK surprisingly inhibits endothelium‐dependent hyperpolarization‐like relaxations in rat mesenteric arteries

Pages: 2905-2921

Article date: August 2019

Authors: Hui Chen, Paul M. Vanhoutte, Susan W.S. Leung

Efficacious dose of metformin for breast cancer therapy is determined by cation transporter expression in tumours

Pages: 2724-2735

Article date: August 2019

Authors: Hao Cai, Ruth S. Everett, Dhiren R. Thakker