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British Journal of Pharmacology

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A novel cyclic biased agonist of the apelin receptor, MM07, is disease modifying in the rat monocrotaline model of pulmonary arterial hypertension

Pages: 1206-1221

Article date: May 2019

Authors: Peiran Yang, Cai Read, Rhoda E. Kuc, Duuamene Nyimanu, Thomas L. Williams, Alexi Crosby, Guido Buonincontri, Mark Southwood, Stephen J. Sawiak, Robert C. Glen, Nicholas W. Morrell, Anthony P. Davenport, Janet J. Maguire

Neprilysin inhibition for pulmonary arterial hypertension: a randomized, double‐blind, placebo‐controlled, proof‐of‐concept trial

Pages: 1251-1267

Article date: May 2019

Authors: Adrian J. Hobbs, Amie J. Moyes, Reshma S. Baliga, Dipa Ghedia, Rachel Ochiel, Yvonne Sylvestre, Caroline J. Doré, Kashfia Chowdhury, Kate Maclagan, Harriet L. Quartly, Reecha Sofat, Angelique Smit, Benjamin E. Schreiber, Gerry J. Coghlan, Raymond J. MacAllister

From identification to functional characterization of cyriotoxin‐1a, an antinociceptive toxin from the spider Cyriopagopus schioedtei

Pages: 1298-1314

Article date: May 2019

Authors: Tânia C. Gonçalves, Evelyne Benoit, Michael Kurz, Laetitia Lucarain, Sophie Fouconnier, Stéphanie Combemale, Lucie Jaquillard, Brigitte Schombert, Jean‐Marie Chambard, Rachid Boukaiba, Gerhard Hessler, Andrees Bohme, Laurent Bialy, Stéphane Hourcade, Rémy Béroud, Michel De Waard, Denis Servent, Michel Partiseti

Modafinil protects hippocampal neurons by suppressing excessive autophagy and apoptosis in mice with sleep deprivation

Pages: 1282-1297

Article date: May 2019

Authors: Yin Cao, Qinglin Li, Lulu Liu, Hui Wu, Fei Huang, Changhong Wang, Yunyi Lan, Fang Zheng, Faping Xing, Qiang Zhou, Qi Li, Hailian Shi, Beibei Zhang, Zhengtao Wang, Xiaojun Wu

Cannabinoid CB1 and CB2 receptor mechanisms underlie cannabis reward and aversion in rats

Pages: 1268-1281

Article date: May 2019

Authors: Krista J. Spiller, Guo‐hua Bi, Yi He, Ewa Galaj, Eliot L. Gardner, Zheng‐Xiong Xi

Evidence for metabotropic function of epithelial nicotinic cholinergic receptors in rat colon

Pages: 1328-1340

Article date: May 2019

Authors: Lena Lottig, Sandra Bader, Marcel Jimenez, Martin Diener

The MC4 receptor agonist RO27‐3225 inhibits NLRP1‐dependent neuronal pyroptosis via the ASK1/JNK/p38 MAPK pathway in a mouse model of intracerebral haemorrhage

Pages: 1341-1356

Article date: May 2019

Authors: Shengpan Chen, Yuchun Zuo, Lei Huang, Prativa Sherchan, Jian Zhang, Zhengtao Yu, Jianhua Peng, Junyi Zhang, Lianhua Zhao, Desislava Doycheva, Fei Liu, John H. Zhang, Ying Xia, Jiping Tang

The impact of dihydropyridine derivatives on the cerebral blood flow response to somatosensory stimulation and spreading depolarization

Pages: 1222-1234

Article date: May 2019

Authors: Írisz Szabó, Orsolya M. Tóth, Zsolt Török, Dániel Péter Varga, Ákos Menyhárt, Rita Frank, Dóra Hantosi, Ákos Hunya, Ferenc Bari, Ibolya Horváth, László Vigh, Eszter Farkas

Novel molecular mechanisms in the inhibition of adrenal aldosterone synthesis: Action of tolvaptan via vasopressin V2 receptor‐independent pathway

Pages: 1315-1327

Article date: May 2019

Authors: Yusuf Ali, Kaoru Dohi, Ryuji Okamoto, Kan Katayama, Masaaki Ito

Semaphorin‐3E attenuates intestinal inflammation through the regulation of the communication between splenic CD11C+ and CD4+CD25 T‐cells

Pages: 1235-1250

Article date: May 2019

Authors: Laëtitia Kermarrec, Nour Eissa, Hongxing Wang, Kunal Kapoor, Abdoulaye Diarra, Abdelilah S. Gounni, Charles N. Bernstein, Jean‐Eric Ghia