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British Journal of Pharmacology

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Short lipopeptides specifically inhibit the growth of Propionibacterium acnes with a dual antibacterial and anti‐inflammatory action

Pages: 2321-2335

Article date: July 2019

Authors: Guang Yang, Jingyu Wang, Shengsheng Lu, Zhao Chen, Sheng Fan, Daiwei Chen, Huanxin Xue, Wenyuan Shi, Jian He

Androgen receptor antagonism accelerates disease onset in the SOD1G93A mouse model of amyotrophic lateral sclerosis

Pages: 2111-2130

Article date: July 2019

Authors: Victoria M. McLeod, Chew L. Lau, Mathew D.F. Chiam, Thusitha W. Rupasinghe, Ute Roessner, Elvan Djouma, Wah C. Boon, Bradley J. Turner

Issue Information

Pages: 2109-2110

Article date: July 2019

VU0810464, a non‐urea G protein‐gated inwardly rectifying K+ (Kir3/GIRK) channel activator, exhibits enhanced selectivity for neuronal Kir3 channels and reduces stress‐induced hyperthermia in mice

Pages: 2238-2249

Article date: July 2019

Authors: Baovi N. Vo, Kristopher K. Abney, Allison Anderson, Ezequiel Marron Fernandez de Velasco, Michael A. Benneyworth, John Scott Daniels, Ryan D. Morrison, Corey R. Hopkins, Charles David Weaver, Kevin Wickman

Inactivation of endothelial adenosine A2A receptors protects mice from cerebral ischaemia‐induced brain injury

Pages: 2250-2263

Article date: July 2019

Authors: Yaqi Zhou, Xianqiu Zeng, Ge Li, Qiuhua Yang, Jiean Xu, Min Zhang, Xiaoxiao Mao, Yapeng Cao, Lina Wang, Yiming Xu, Yong Wang, Yu Zhang, Zhengshuang Xu, Chaodong Wu, Jiang‐Fan Chen, Md Nasrul Hoda, Zhiping Liu, Mei Hong, Yuqing Huo

Analgesic transient receptor potential vanilloid‐1‐active compounds inhibit native and recombinant T‐type calcium channels

Pages: 2264-2278

Article date: July 2019

Authors: Jeffrey R. McArthur, Rocio K. Finol‐Urdaneta, David J. Adams

Action of MK‐7264 (gefapixant) at human P2X3 and P2X2/3 receptors and in vivo efficacy in models of sensitisation

Pages: 2279-2291

Article date: July 2019

Authors: David Richards, Joel R. Gever, Anthony P. Ford, Samuel J. Fountain

Oral administration of a new HRI activator as a new strategy to improve high‐fat‐diet‐induced glucose intolerance, hepatic steatosis, and hypertriglyceridaemia through FGF21

Pages: 2292-2305

Article date: July 2019

Authors: Mohammad Zarei, Eugènia Pujol, Tania Quesada‐López, Francesc Villarroya, Emma Barroso, Santiago Vázquez, Javier Pizarro‐Delgado, Xavier Palomer, Manuel Vázquez‐Carrera

Amlodipine induces vasodilation via Akt2/Sp1‐activated miR‐21 in smooth muscle cells

Pages: 2306-2320

Article date: July 2019

Authors: Qin Fang, Min Tian, Feng Wang, Zhihao Zhang, Tingyi Du, Wei Wang, Yong Yang, Xianqing Li, Guangzhi Chen, Lei Xiao, Haoran Wei, Yan Wang, Chen Chen, Dao Wen Wang

Cyclic nucleotide signalling compartmentation by PDEs in cultured vascular smooth muscle cells

Pages: 1780-1792

Article date: June 2019

Authors: Liang Zhang, Kaouter Bouadjel, Boris Manoury, Grégoire Vandecasteele, Rodolphe Fischmeister, Véronique Leblais

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